Peroxisome proliferator-activated receptor δ (PPARδ) stimulation or over-expression in adipocytes leads to increased fatty acid oxidation, improved exercise tolerance, and resistance to obesity. GW 501516 is the first highly selective synthetic PPARδ agonist available. GW 501516 binds to human PPARδ with an IC50 value of 1 nM, and is at least 100-fold selective for PPARδ compared to PPARα and PPARγ. In obese primates, GW 501516 increases high density lipoprotein cholesterol and apolipoprotein A-1 specific reverse cholesterol transport. GW 501516 is therefore a model compound for a new type of obesity therapeutic, as well as a selective pharmacological tool for understanding lipid metabolism.
| GW-501516 Chemical Properties |
| Melting point |
134-136°C |
| Boiling point |
584.5±60.0 °C(Predicted) |
| density |
1.42±0.1 g/cm3(Predicted) |
| storage temp. |
-20°C |
| solubility |
DMSO: soluble20mg/mL, clear |
| form |
powder |
| pka |
3.17±0.10(Predicted) |
| color |
white to beige |
| BRN |
18515150 |
| Stability: |
Light Sensitive |
What is Cardarine?
Cardarine, also referred to as GW501516, is a synthetic compound that serves as a metabolic modulator.
People often think it’s a type of compound called a SARM (selective androgen receptor modulator), but Cardarine actually belongs to a class of drugs called peroxisome proliferator-activated receptor (PPAR) agonists.
The cell receptors these affect are most abundant in muscle cells throughout the body.
Compounds such as Cardarine act upon energy metabolism in the cells and are thought to increase energy expenditure.
This is why some athletes and bodybuilders are attracted to taking Cardarine. They may take it in hopes of increasing fat-burning, getting a leaner body composition, and increasing their sport performance.
Benefits of Using Cardarine GW-501516
Even though there are lots of negative effects of injecting Cardarine, there are some benefits as well, due to which it has gained such high popularity among the masses. The various advantages of using this drug include:
● Increase in endurance
● Better Fat burning
● Improve the performance of Athletes
Side effects of Cardarine GW-501516
There are not just one but multiple side effects of using this synthetic SARM. Even though people use this product, it is not as safe as various websites or reviews claim. If you wish to use a product, you must read and understand everything about its use case and make an informed decision afterward.
Not just abuse, addiction, or overdose; there is much more that Cardarine GW-501516 does to your body.
● High chances of developing Cancer
● Damages the Brain
● Severe Headache
● Messes with the cardiovascular system
● Muscle Cramps and Joint Pains
● Damages the Liver
● Stomach Upset
